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  6. 11913610MG

MilliporeSigma™ Calbiochem™ Adenosine A1 Receptor Agonist II, CCPA

Catalog No. 11913610MG Shop All MilliporeSigma Products
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10mg

Description

An adenosine analog that acts as a selective, high affinity agonist for Adenosine A1 receptor (A1R) (Ki = 800 pM

An adenosine analog that acts as a selective, high affinity agonist for Adenosine A1 receptor (A1R) (Ki = 800 pM; 2.3μM, 18.8μM, and 42nM for human A1, A2A, A2B, A3 respectively). Shown to be centrally active following systemic administration and exhibits anti-convulsive effects. Also reported to inhibit adenylate cyclase activity in rat fat cell membrane (IC50 = 33nM). Diminishes respiratory rhythm, reduces heart rate, and enhances the activity of KATP channels. Reduces norepinephrine release by about 50% in untreated and pertussis toxin treated hearts.

Specifications

Form Solid
Content And Storage Protect from light
Quantity 10 mg
Color White
Description 99% by HPLC
Target Proteins A1
Molecular Formula C15H20ClN5O4
Formula Weight 369.8g/mol
Solubility DMSO or H2O
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