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MilliporeSigma™ Calbiochem™ SB-277011-A Dihydrochloride

Catalog No. 5054840001 Shop All MilliporeSigma Products
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5mg

Description

A brain-penetrant, high-affinity, and selective dopamine D3 receptor antagonist

A brain-penetrant, high-affinity, and selective dopamine D3 receptor antagonist. High affinity for the hD3 receptor (pKi = 7.95) with 100-fold selectivity over the hD2 receptor and over 66 other receptors, enzymes, and ion channels. Rat data shows that the compound is selective for the D3 receptor over certain serotonergic and cholinergic receptors at doses up to 56.0mg/kg and strong physiological response at 32.0mg/kg.

Specifications

Quantity 5 mg
Form Solid
Content And Storage Hygroscopic, Protect from light
Color White
Description 98% by HPLC
Target Proteins D3
Molecular Formula C28H30N4O·2HCl
Solubility H2O
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