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  8. PD 81723, Tocris Bioscience™

PD 81723, Tocris Bioscience™

Catalog No. p-4785325 Shop All R&D Systems Products
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Quantity:
10 mg
50 mg
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Description

Allosteric potentiator of A1 receptors

Allosteric potentiator at the adenosine A1 receptor; acts via agonist-dependent and -independent mechanisms. Enhances agonist affinity for, and increased t½ of dissociation from, the receptor. Also inhibits basal and forskolin-stimulated adenylyl cyclase (AC) activity in A1 receptors expressed in CHO cells, possibly via direct potentiation of constitutive receptor activity or by direct inhibition of AC. Active in vivo.

Chemical Identifiers

CAS 132861-87-1
Molecular Formula C14H12F3NOS
Molecular Weight (g/mol) 299.311
InChI Key KKDKAWKYGCUOGR-UHFFFAOYSA-N
Synonym 2-amino-4,5-dimethylthiophen-3-yl 3-trifluoromethyl phenyl methanone, 2-amino-4,5-dimethyl-3-thienyl-3-trifluoromethyl phenyl methanone, chembl59532, 2-amino-4,5-dimethylthiophen-3-yl-3-trifluoromethyl phenyl methanone, methanone, 2-amino-4,5-dimethyl-3-thienyl 3-trifluoromethyl phenyl, 4,5-dimethyl-3-3-trifluoromethyl benzoyl thiophen-2-amine, tocris-1363, d07hxl
PubChem CID 122028
IUPAC Name (2-amino-4,5-dimethylthiophen-3-yl)-[3-(trifluoromethyl)phenyl]methanone
SMILES CC1=C(SC(=C1C(=O)C2=CC(=CC=C2)C(F)(F)F)N)C

Specifications

Quantity 10 mg
Formula Weight 299.31
Percent Purity >99%
Chemical Name or Material PD 81723

Safety and Handling

Recommended Storage Store at Room Temperature
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