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  7. Sumanirole maleate, Tocris Bioscience™

Sumanirole maleate, Tocris Bioscience™

Catalog No. 277350 Shop All R&D Systems Products
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Quantity:
10 mg
50 mg
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This item is not returnable. View return policy

Description

Selective D2 agonist

High affinity D2 receptor agonist (EC50 values are between 17 and 75 nM in cell-based assays). Originally reported to exhibit >200-fold selectivity for the D2 receptor versus other dopamine receptor subtypes (Ki values are 9.0, 1940, >2190 and >7140 for D2, D3, D4 and D1 receptors respectively). More recently reported to be around 32-fold selective for D2 over D3 receptors (Ki values are 17.1 and 546 nM respectively). Exhibits antiParkinsonian activity.

Chemical Identifiers

CAS 179386-44-8
Molecular Formula C15H17N3O5
Molecular Weight (g/mol) 319.317
InChI Key VOJRMYBBPKNLLI-ORHWHDKWSA-N
Synonym sumanirole maleate, unii-2oi87t3r1b, u 95666e sumanirole maleate, r-5,6-dihydro-5-methylamino-4h-imidazo 4,5,1-ij quinolin-2 1h-one z-2-butenedioate, u 95666e, sumanirole maleate, r-5,6-dihydro-5-methylamino-4h-imidazo 4,5,1-ij quinolin-2 1h-one 2z-2-butenedioate, maleate, sumanirole maleate hplc, 5,6-dihydro-5-methylamino-4h-imidazo 4,5,1-ij quinolin-2 1h-one, r-maleate
PubChem CID 9818478
SMILES CNC1CC2=C3C(=CC=C2)NC(=O)N3C1.C(=CC(=O)O)C(=O)O

Specifications

Quantity 50 mg
Formula Weight 319.31
Percent Purity >98%
Chemical Name or Material Sumanirole maleate

Safety and Handling

Recommended Storage Store at -20°C
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