Benzoxazines
Benzoxazines
TARGETMOL CHEMICALS INC PRIDOPIDINE 10MG
Also available in 2 mg 5 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Pridopidine (FR310826) a dopamine (DA) stabilizer acts as a low affinity dopamine D2 receptor (D2R) antagonist improves motor performance and shows neuroprotective effects in Huntington disease R6/2 mouse model. purity: 99%
TARGETMOL CHEMICALS INC ABAPERIDONE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg and bulk. Please contact Fisher for quotes. Abaperidone is a potent 5-HT2A receptor and dopamine D2 receptor antagonist with an IC50 of 6.2 for 5-HT2A receptors and 17 nM for dopamine D2 receptors.Abaperidone is a potentially atypical anti-psychotropic compound that reduces basal hsp70 mRNA expression in rat striatum and prefrontal cortex. expression in the striatum and prefrontal cortex of rats. purity: 94%
TARGETMOL CHEMICALS INC SAFINAMIDE 5MG
Also available in 10 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Safinamide (FCE-26743) is a reversible and selective monoamine oxidase B (IC50 0.098uM) inhibitor reducing the degradation of dopamine and a glutamate release inhibitor (IC50 8uM). It also inhibits dopamine reuptake. Safinamide also blocks sodium and calcium channels. Potential additional uses of Safinamide might be Parkinson's disease restless leg syndrome and epilepsy. purity: 99%
TARGETMOL CHEMICALS INC ROTIGOTINE 5MG
Also available in 10mg 25mg 50mg 100mg and bulk. Please contact Fisher for quotes. Rotigotine (1-Naphthalenol 5678-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist. purity: 99%
TARGETMOL CHEMICALS INC ROTUNDINE 500MG
Also available in 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Rotundine (Gindarine) (L-tetrahydropalmatine L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM. purity: 99%
TARGETMOL CHEMICALS INC VANOXERINE DIHYDROCHLORI 50MG
Also available in 5 mg 10 mg 25 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 1-51 nM)purity: 97%
TARGETMOL CHEMICALS INC SYROSINGOPINE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Syrosingopine has selective depleting effect on brain amines is potentiated by combined treatment with disulfiram or fusaric acid a dopamine beta-hydroxylase inhibitor. purity: 99%
TARGETMOL CHEMICALS INC HALOPEMIDE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2). Halopemid is an antagonist of dopamine receptors. Halopemid can be used in psychotropic research. purity: 96%
TARGETMOL CHEMICALS INC SERTINDOLE 25MG
Also available in 5 mg 10 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Sertindole (Lu 23-174) is an atypical antipsychotic that binds to dopamine D2 receptors and the serotonin (5-HT) receptor subtypes 5-HT1D 5-HT2A and 5-HT2C (Kds = 2.7 20 0.14 and 6 nM respectively)purity: 99%
TARGETMOL CHEMICALS INC AMPEROZIDE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Amperozide (FG 5606) is a diphenylbutylpiperazine atypical antipsychotic which antagonizes 5-HT2A receptors. It inhibits dopamine release and alters the firing of dopaminergic neurons. Investigations regarding the use of the agent revolved primarily around its capability for treating schizophrenia in humans. purity: 99%
TARGETMOL CHEMICALS INC ORDOPIDINE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg and bulk. Please contact Fisher for quotes. Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity. Ordopidine acts as a dopamine D2 receptor antagonist in vitro and despite its low affinity its specific state-dependent behavioral effect characteristics are not generally shared by D2 receptor antagonists. purity: 99%
TARGETMOL CHEMICALS INC CABERGOLINE 10MG
Also available in 1 mg 5 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Cabergoline (FCE-21336) is an ergot derived-dopamine D2-like receptor agonist. It has high affinity for D2 D3 and 5-HT2B receptors (Ki=0.7 1.5 and 1.2 respectively).Cabergoline permits rapid and effective hormonal and tumor control by normalizing prolactin-producing pituitary adenomas levels. purity: 99%
TARGETMOL CHEMICALS INC ROTIGOTINE- 25MG
Also available in 5 mg 10 mg 50 mg 100 mg 200 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome. Administered as a once-daily transdermal patch Rotigotine has not been associated with serum enzyme elevations during treatment or with episodes of clinically apparent liver injury. purity: 99%
TARGETMOL CHEMICALS INC ECOPIPAM 5MG
Also available in 1 mg 2 mg 10 mg 25 mg 50 mg and bulk. Please contact Fisher for quotes. Ecopipam (UNII-0X748O646K) is a potent selective and orally active antagonist of dopamine D1/D5 receptor with Kis of 1.2 nM and 2.0 nM respectively. Ecopipam shows more than 40-flod selectivity over D2 D4 5-HT and (alpha)2a receptor (Ki=0.98 5.52 0.08 and 0.73 uM respectively). Ecopipam can be used for the research of schizophrenia and obesity. purity: 98%
TARGETMOL CHEMICALS INC 6-CHLOROMELATONIN 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg and bulk. Please contact Fisher for quotes. 6-Chloromelatonin is a potent melatonin receptor agonist a 5-methoxyindole compound that competes for the same presynaptic melatonin receptor sites in the rabbit retina and inhibits the calcium-dependent release of [3H]dopamine with a higher metabolic stability than melatonin. Chloromelatonin competes for [3H]melatonin binding to MT2 receptors (pKi=9.77) and may be used to study insomnia and sleep disorders associated with depression. purity: 99%
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