Cayman Chemical PovIdon-IodIn 25g
An agonist of the dopamine D1 receptor (Ki40 nM) induces activity equal to or greater than dopamine in fish retinas and rat caudate-putman (EC50s 7 4 and 1 1 nM respectively) does not show agonist behavior for the D2 receptor expressed in MMQ cells ( 10 M) induces desensitization of dopamine-stimulated cAMP accumulation and reduces D1 receptor expression by 79 in C-6 glioma cells expressing monkey D1A receptors (10 M) increases locomotor activity 5 3-fold and reduces disease severity in a MPTP-treated marmoset model of Parkinsons disease (3 mol/kg s c ) elicits over a 230 increase in cortical and hippocampal acetylcholine release (4 mol/kg s c )