Lysates
Cayman Chemical BLT1 Receptrmouse Monclo 100ug
A dopamine D1 receptor agonist (K0 5 4 nM in a radioligand binding assay) selective for dopamine D1 over D2 receptors (K0 5 73 nM) induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striatal membranes (EC50 491 nM) prevents and reverses fentanyl-induced respiratory depression in cats at 3 mg/kg increases locomotion and rearing in rats
Cayman Chemical 1 3DIpalmItoleoyl Glycerol 1mg
A histamine H1 receptor antagonist selective over H3 a1- a2- andBadrenergic dopamine D2long serotonin 5-HT2 muscarinic acetylcholine and benzodiazepine receptors reduces dye leakage from the nasal passages of sensitized rats (ED50 0.03 mg/kg) inhibits histamine-induced bronchoconstriction in the anesthetized dog (ED50 3.2 Ug/kg) dose-dependently prevents conjunctival vascular hyperpermeability a in guinea pig model of conjunctivitis
Cayman Chemical IgMhumn Monclonal ntIbo 100ug
An agonist of a4B2 subunit-containing nAChRs (Ki 43 pM) selective for a4B2 subunit-containing nAChRs over a7 nAChRs (Ki 230 nM) 86Rb flux in IMR-32 cells (EC50 7 nM) induces dopamine release from rat striatal slices (EC50 0.4 nM) induces analgesia in the hot plate test and the Straub-tail response in mice (ED50s 0.005 and 0.02 mg/kg respectively)
Cayman Chemical τ-FluvalInate 100mg
An agonist of nicotinic AChRs selective for a4B2 or a7 subunit-containing nicotinic AChRs (Kis 0.7 and 10.9 nM in isolated rat cortex and isolated rat hippocampus respectively) over a1Bɣ subunit-containing nicotinic AChRs (EC50 1000 nM in PC12 cells) induces dopamine release from isolated rat striatal synaptosomes (EC50 2.4 nM) and increases nicotine-induced elevations in epinephrine and norepinephrine levels in isolated rat adrenal gland at 100 UM inhibits nicotine-induced ion flux in isolated rat thalamic synaptosomes (IC50 154 nM)